Enerion, pills 200mg 60pcs

Composition

1 coated tablet contains:

Active ingredient:

sulbutyamine 200 mg;

Auxiliary substances:

corn starch-12 mg;

dried starch paste-40 mg;

glucose (dextrose) anhydrous-20 mg;

lactose monohydrate-65.5 mg;

magnesium stearate-3.5 mg;

talc-9 mg;

Shell:

sodium bicarbonate — 0,603 mg; sodium carboxymethylcellulose — 0,556 mg; white beeswax — 0,201 mg; titanium dioxide (E171) — of 8.43 mg; ethyl cellulose — appears to be 0.485 mg; sunset yellow (Sunset yellow FCF, E110) — 3 mg; glycerol monooleate — 0,242 mg; Polysorbate 80 — 0,302 mg; povidone — 0,692 mg; sucrose — 106,956 mg; silicon dioxide colloidal anhydrous (Aerosil 130) — 0,404 mg, talc — 28,21 mg

Pharmacological action

The drug Enerion is a synthetic compound similar in structure to thiamine, in comparison with which the molecule has an open thiazole cycle, an additional disulfide bond, and a lipophilic ether.

Due to this modification, sulbutyamine is highly soluble in fats, is quickly absorbed from the gastrointestinal tract and easily penetrates the BBB; unlike thiamine, it can accumulate in the cells of the reticular formation, hippocampus and dentate gyrus, as well as Purkinje cells and glomeruli of the granular layer of the cerebellar cortex.

While taking Enerion, coordination of movement improves and resistance to physical exertion increases, and the resistance of the cerebral cortex structures to repeated anoxia increases. The drug is effective in the symptomatic treatment of functional asthenia.

Pharmacokinetics

Sulbutyamine is rapidly absorbed, _{and cmax} of the drug in blood plasma is reached 1-2 hours after use. T_1/2 — about 5 hours. The drug is excreted in the urine.

Indications

Symptomatic treatment of functional asthenia.

Use during pregnancy and lactation

According to the results of clinical studies, the drug does not affect the development of the fetus.

However, due to the lack of sufficient clinical data, Enerion is not recommended for use during pregnancy, as well as during breast-feeding, as it is currently unknown whether sulbutyamine is able to enter breast milk.

Contraindications

Hypersensitivity to any of the components of Enerion.

With caution: persons under 18 years of age (the drug is not recommended to be prescribed due to the lack of clinical data).

Side effects

Allergic reactions (the presence of Sunset yellow dye in the preparation), digestive disorders, neuropsychiatric reactions (tremor, headache, agitation, general malaise).

How to take, course of use and dosage

Inside. Enerion is recommended for use only in adult patients.

The daily dose is 2-3 tablets (400-600 mg) in 2 divided doses (during breakfast and lunch).

The duration of treatment should not exceed 4 weeks.

Overdose

Symptoms: agitation with euphoria and tremor of the extremities are transient in nature and do not require special treatment.

Special instructions

The excipients of Enerion include lactose monohydrate.

As a result, this drug is not recommended for people with lactose deficiency, galactosemia, or glucose/galactose malabsorption syndrome.

Influence on the ability to drive a car and perform work that requires a high rate of psychomotor reactions. It doesn’t affect you.

Form of production

Tablets

Storage conditions

At a temperature not exceeding 25 °C

Shelf life

3 years

Active ingredient

Sulbutyamine

Dosage form

Tablets

Description

For adults as directed by your doctor

Indications

Asthenia